GTX-758
Based on 1 Customer Validation
GTX-758 is an orally active, nonsteroidal, selective agonist of ERα. GTX-758 plays an important role in castration resistant prostate cancer (CRPC) research.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 純度 : 99.59%
- CAS 番号: 938067-78-8
- 分子式: C19H13F2NO3
- 分子量:341.31
-
保管条件:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
生物活性
-
化学情報
-
溶剤 & 溶解度
- 純度とドキュメンテーション
- 参考文献
-
Help & FAQs
生物活性
製品説明
IC50 & Target
|
ERα |
臨床実験
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
化学情報
-
CAS 番号 938067-78-8
-
性状 Solid
-
分子量 341.31
-
分子式 C19H13F2NO3
-
Color White to off-white
-
SMILES
O=C(N(C1=CC=C(F)C=C1)C2=CC=C(O)C=C2)C3=CC=C(O)C(F)=C3
-
別名
Capesaris
-
輸送条件
Room temperature in continental US; may vary elsewhere.
-
保管条件
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
溶剤 & 溶解度
体外:
DMSO : 100 mg/mL (292.99 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
純度とドキュメンテーション
-
データシート (282 KB)
-
SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
-
取扱説明書 (2659 KB)
参考文献
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.9299 mL | 14.6494 mL | 29.2989 mL | 73.2472 mL |
| 5 mM | 0.5860 mL | 2.9299 mL | 5.8598 mL | 14.6494 mL | |
| 10 mM | 0.2930 mL | 1.4649 mL | 2.9299 mL | 7.3247 mL | |
| 15 mM | 0.1953 mL | 0.9766 mL | 1.9533 mL | 4.8831 mL | |
| 20 mM | 0.1465 mL | 0.7325 mL | 1.4649 mL | 3.6624 mL | |
| 25 mM | 0.1172 mL | 0.5860 mL | 1.1720 mL | 2.9299 mL | |
| 30 mM | 0.0977 mL | 0.4883 mL | 0.9766 mL | 2.4416 mL | |
| 40 mM | 0.0732 mL | 0.3662 mL | 0.7325 mL | 1.8312 mL | |
| 50 mM | 0.0586 mL | 0.2930 mL | 0.5860 mL | 1.4649 mL | |
| 60 mM | 0.0488 mL | 0.2442 mL | 0.4883 mL | 1.2208 mL | |
| 80 mM | 0.0366 mL | 0.1831 mL | 0.3662 mL | 0.9156 mL | |
| 100 mM | 0.0293 mL | 0.1465 mL | 0.2930 mL | 0.7325 mL |
GTX-758 関連分類
HY-111061 関連分類
Powered by Bioz