MOR agonist-4
MOR agonist-4 (2d) is a G protein signaling-biased Kappa opioid receptor (KOR) agonist with an EC50 value of 11 nM. MOR agonist-4 contains an electron withdrawing CF3 group and a bias factor of 38 based on triazole. MOR agonist-4 is used in the research of pruritis and analgesia.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 3050669-97-8
- 分子式: C22H19F3N4S
- 分子量:428.47
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
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生物活性
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化学情報
- 純度とドキュメンテーション
- 参考文献
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Opioid Receptor アイソフォーム固有の製品をすべて表示
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生物活性
製品説明
体外実験
MOR agonist-4 (10 μM) completely inhibits U69,593 binding of an appropriate radiolabeled receptor ligand to KOR with a Ki value of 5.8 nM, but binding of ligands to MOR and DOR is poorly inhibited (30.9 % and 30.7 %, respectively)[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only. .
化学情報
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CAS 番号 3050669-97-8
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分子量 428.47
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分子式 C22H19F3N4S
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SMILES
CC(C=C1)=C(C(F)(F)F)C=C1CCC(N2CC3=CC=CS3)=NN=C2C4=CC=CC=N4
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
MOR agonist-4 関連分類
HY-161812 関連分類
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