M4R ligand-1
M4R ligand-1 is a M4R ligand. M4R ligand-1 binds to the extracellular vestibular allosteric site of M4R. M4R ligand-1 can be used for the research of schizophrenia.
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- Formel: C24H24N4O3
- Molecular Weight:416.47
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biologische Aktivität
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Chemical Information
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Help & FAQs
Biologische Aktivität
Beschreibung
IC50 & Target
[1]|
mAChR4 |
In Vitro
M4R ligand-1 (MKcpd-97(2)) is a positive allosteric modulator of M4R; when combined with ACh, its allosteric site affinity pKB is 6.50; when combined with Xanomeline (HY-105182), the corresponding allosteric site affinity pKB is 6.14[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Molecular Weight 416.47
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Formel C24H24N4O3
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SMILES
CN1C(C2=CC(C3=NC(C(O)=O)=CC=C3C4=CN(N=C4)CC5CCCC5)=CC=C2C1)=O
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
M4R ligand-1 Related Classifications
HY-189040 Related Classifications
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