Mutant IDH1-IN-3
Mutant IDH1-IN-3 (Compound 1) is a selective allosteric inhibitor of mutant isocitrate dehydrogenase 1 (IDH1). Mutant IDH1-IN-3 has an IC50 of 13 nM for R132H IDH1. Mutant IDH1-IN-3 inhibits the production of D-2-hydroxyglutaric acid (2HG) in cells. Mutant IDH1-IN-3 can be used in the study of cancer.
For research use only. We do not sell to patients.
- CAS No.: 1648909-73-2
- Formula: C22H30N4O
- Molecular Weight:366.50
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
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Help & FAQs
Biological Activity
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R132H IDH1 13 nM (IC50) |
Chemical Information
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CAS No. 1648909-73-2
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Molecular Weight 366.50
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Formula C22H30N4O
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SMILES
OC1=C(CN2C=CN=C2)C=C(C(C)(C)CC(C)(C)C)C=C1CN3C=CN=C3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Mutant IDH1-IN-3 Related Classifications
HY-100476 Related Classifications
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