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  3. N-desmethyl Enzalutamide D6

N-desmethyl Enzalutamide D6 (Synonyms: N-desmethyl MDV 3100 D6)

Cat. No.: HY-70002AS
Handling Instructions

N-desmethyl Enzalutamide D6 (N-desmethyl MDV 3100 D6) is a deuterium labeled N-desmethyl Enzalutamide. N-desmethyl Enzalutamide is an active metabolite of Enzalutamide. N-desmethyl Enzalutamide is the active metabolite of Enzalutamide. N-desmethyl Enzalutamide demonstrates primary and secondary pharmacodynamics of similar potency to Enzalutamide and circulates at approximately the same plasma concentrations as enzalutamide.

For research use only. We do not sell to patients.

N-desmethyl Enzalutamide D6 Chemical Structure

N-desmethyl Enzalutamide D6 Chemical Structure

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Description

N-desmethyl Enzalutamide D6 (N-desmethyl MDV 3100 D6) is a deuterium labeled N-desmethyl Enzalutamide. N-desmethyl Enzalutamide is an active metabolite of Enzalutamide. N-desmethyl Enzalutamide is the active metabolite of Enzalutamide. N-desmethyl Enzalutamide demonstrates primary and secondary pharmacodynamics of similar potency to Enzalutamide and circulates at approximately the same plasma concentrations as enzalutamide[1].

IC50 & Target

Androgen-receptor[1]

Molecular Weight

456.45

Formula

C₂₀H₈D₆F₄N₄O₂S

SMILES

S=C(N1C2=CC(F)=C(C(N)=O)C=C2)N(C3=CC=C(C(C(F)(F)F)=C3)C#N)C(C(C([2H])([2H])[2H])1C([2H])([2H])[2H])=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

N-desmethyl Enzalutamide D6N-desmethyl MDV 3100 D6Androgen ReceptorDeuteriumlabeledmetaboliteEnzalutamidepharmacodynamicscirculatesCYP2C8CYP3A4Inhibitorinhibitorinhibit

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N-desmethyl Enzalutamide D6
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HY-70002AS
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