Picumeterol
Picumeterol (GR114297A) is a potent and selective β2-adrenoceptor agonist with bronchodilator and anti-bronchoconstrictor effects. Picumeterol produces long-lasting relaxation of airways smooth muscle both in vitro and in vivo. Picumeterol is cleared from plasma through a rapid and extensive hepatic metabolism. Picumeterol is proming for rasearch of asthma and related diseases.
For research use only. We do not sell to patients.
- CAS No.: 130641-36-0
- Formula: C21H29Cl2N3O2
- Molecular Weight:426.38
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Adrenergic Receptor Isoforms
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Biological Activity
Chemical Information
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CAS No. 130641-36-0
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Molecular Weight 426.38
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Formula C21H29Cl2N3O2
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SMILES
O[C@H](C1=CC(Cl)=C(C(Cl)=C1)N)CNCCCCCCOCCC2=CC=CC=N2
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Synonyms
GR114297A
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
[1]. Weersink EJ, et al. Picumeterol: dissociation of improvement in lung function and reduction of airways hyperresponsiveness in asthmatics. Br J Clin Pharmacol. 1997 Feb;43(2):169-76. [Content Brief]
[2]. Barrow A, et al. Kinetics and disposition of picumeterol in animals. Xenobiotica. 1995 Sep;25(9):993-1007. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)