PIN1 degrader-2
PIN1 degrader-2 (compound 164A10) is a potent and selective covalent PIN1 degrader (IC50 = 4.1 nM) that induces PIN1 degradation in cancer cells (DC50 < 500 nM). PIN1 degrader-2 can be used for cancer research.
For research use only. We do not sell to patients.
- CAS No.: 3080918-74-4
- Formula: C31H32ClFN6O4
- Molecular Weight:607.07
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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PIN1 4.1 nM (IC50) |
Chemical Information
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CAS No. 3080918-74-4
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Molecular Weight 607.07
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Formula C31H32ClFN6O4
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SMILES
NC([C@H](CC1=CNC2=C1C=C(F)C=C2)NC([C@@H]3CCCCN3C([C@@H]4CC5=C(CN4C(CCl)=O)NC6=C5C=CC=C6)=O)=O)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)