From 4,5,6,7-tetrahydro-5-methylimidazo[4,5,1-jk](1,4)benzodiazepin-2(1H)-one (TIBO) to etravirine (TMC125): fifteen years of research on non-nucleoside inhibitors of HIV-1 reverse transcriptase
- J Med Chem. 2005 Mar 24;48(6):1689-96. doi: 10.1021/jm040127p.
Affiliations
- 1. Drug Discovery, Johnson & Johnson Pharmaceutical Research & Development, Welsh and McKean Roads, Spring House, Pennsylvania 19477-0776, USA. [email protected]
PMID: 15771411
DOI: 10.1021/jm040127p