Targeted Covalent Inhibition: A Prospective Way to Develop Novel HSP90 C-terminal Inhibitor

  • Curr Drug Targets. 2022;23(16):1454-1456. doi: 10.2174/1389450123666220920111841.
Yajun Liu  1 ,  Yajing Li  1
Affiliations
  • 1. School of Life and Pharmaceutical Sciences, Dalian University of Technology, Dagong Road 2, Liaodongwan District, Panjin 124221, China.
PMID: 36125840 DOI: 10.2174/1389450123666220920111841
Keywords
C-terminus; HSP90; L-cysteine; heat shock response; structure-based drug design; targeted covalent inhibition.
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