Rivulariapeptolides 988
Rivulariapeptolides 988 is a high potent and selective serine protease inhibitor with IC50 values of 95.46 nM, 15.29 nM and 85.50 nM for chymotrypsin, elastase and proteinase K, respectively.
For research use only. We do not sell to patients.
- Formula: C50H68N8O13
- Molecular Weight:989.12
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
IC50: 95.46 nM (chymotrypsin); 15.29 nM (elastase) and 85.50 nM (proteinase K)[1].
Rivulariapeptolides 998 (0-3 μM, 40 min) has high potency and distinct selectivity with IC50 values of 95.46 nM, 15.29 nM and 85.50 nM for chymotrypsin, elastase and proteinase K, respectively[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Molecular Weight 989.12
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Formula C50H68N8O13
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SMILES
CCCC(N1[C@H](C(N[C@H](C(N[C@H](C(N/C(C(N[C@H]2CC[C@@H](O)[N@@]3C2=O)=O)=C\C)=O)[C@@H](C)OC([C@H](C(C)C)NC([C@H](CC4=CC=C(O)C=C4)N(C([C@@H]3CC5=CC=CC=C5)=O)C)=O)=O)=O)[C@H](O)C)=O)CCC1)=O
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Structure Classification
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Initial Source
Cyanobacteria
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)