![[Pyr1]-Apelin-13](https://file.medchemexpress.com/product_pic/hy-p1033.gif "Click to View [Pyr1]-Apelin-13 Product Detail")
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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
11 Results for "
Apelin13
" in MedChemExpress (MCE) Product Catalog:
Products (11)
11 Results for "Apelin13" in MCE Product Catalog:
10
10 Publications Verification
Cat. No.: HY-P1944
CAS No.: 217082-58-1
Target:
10
10 Publications Verification
Cat. No.: HY-P1944A
Target:
10
10 Publications Verification
Target:
연구분야:
ML221 is a potent apelin (APJ) functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in the β-arrestin assay, and EC80 of 10 nM in both assays.
5
Target:
연구분야:
Target:
연구분야:
BMS-986224 is a potent, selective and orally active APJ receptor agonist (Kd = 0.3 nM). BMS-986224 exhibits similar receptor binding and signaling profile to (Pyr 1) apelin-13. BMS-986224 has the potential for the research of heart failure .
Cat. No.: HY-P3162A
Target:
연구분야:
Cat. No.: HY-P1033S1
Target:
연구분야:
Cat. No.: HY-133036
CAS No.: 2287153-38-0
Target:
연구분야:
APJ receptor agonist 1, a biphenyl acid derivative, is a potent APJ receptor (APJ-R) agonist (EC50s 0.093 and 0.12 nM for human and rat APJ-R, respectively). APJ receptor agonist 1 displays in vitro potency to apelin-13, the endogenous peptidic ligand for the APJ receptor. APJ receptor agonist 1 has the potential for the research of heart failure .
Cat. No.: HY-P3162
CAS No.: 568565-11-7
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연구분야:
Cat. No.: HY-P1033S
Target:
연구분야:
Cat. No.: HY-103254R
CAS No.: 877636-42-5
연구분야:
ML221 (Standard) is the analytical standard of ML221 (HY-103254). This product is intended for research and analytical applications. ML221 is a potent apelin (APJ) functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in the β-arrestin assay, and EC80 of 10 nM in both assays.
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
