6 Results for "

CYT387

" in MedChemExpress (MCE) Product Catalog:
Products (6)

6 Results for "CYT387" in MCE Product Catalog:

18
18 Publications Verification
Cat. No.: HY-10961
CAS No.: 1056634-68-4
Purity:  99.37%
Synonyms: CYT387
Target:  

JAK Autophagy Apoptosis

Research Areas:  

Cancer

Momelotinib (CYT387) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50a of 11 nM and 18 nM,respectively. CYT387 shows much less activity against JAK3.
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18
18 Publications Verification
Cat. No.: HY-10962
CAS No.: 1056636-06-6
Purity:  98.06%
Synonyms: CYT387 sulfate salt
Target:  

JAK Autophagy Apoptosis

Research Areas:  

Cancer

Momelotinib sulfate (CYT387 sulfate salt) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50 of 11 nM/18 nM, 10-fold selectivity versus JAK3 (IC50=155 nM).
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Cat. No.: HY-10963
CAS No.: 1056636-07-7
Synonyms: CYT387 mesylate
Target:  

JAK Autophagy

Research Areas:  

Cancer

Momelotinib mesylate (CYT387 mesylate) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50 of 11 nM/18 nM, appr 10-fold selectivity versus JAK3.
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Cat. No.: HY-10961R
CAS No.: 1056634-68-4
Synonyms: CYT387 (Standard)
Research Areas:  

Cancer

Momelotinib (Standard) is the analytical standard of Momelotinib. This product is intended for research and analytical applications. Momelotinib (CYT387) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50a of 11 nM and 18 nM,respectively. CYT387 shows much less activity against JAK3.
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Cat. No.: HY-10961S8
CAS No.: 2056097-81-3
Synonyms: CYT387-d4 hydrochloride hydrate
Momelotinib-d4 (CYT387-d4) dihydrochloride hydrate is a deuterium labeled Momelotinib (HY-10961). Momelotinib (CYT387) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50s of 11 nM and 18 nM,respectively. CYT387 shows much less activity against JAK3 .
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Cat. No.: HY-10962R
CAS No.: 1056636-06-6
Synonyms: CYT387 sulfate salt (Standard)
Research Areas:  

Cancer

Momelotinib (sulfate) (Standard) is the analytical standard of Momelotinib (sulfate). This product is intended for research and analytical applications. Momelotinib sulfate (CYT387 sulfate salt) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50 of 11 nM/18 nM, 10-fold selectivity versus JAK3 (IC50=155 nM).
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