14 Results for "

SSTR4

" in MedChemExpress (MCE) Product Catalog:
Products (14)

14 Results for "SSTR4" in MCE Product Catalog:

Cat. No.: HY-139347
CAS No.: 1638588-92-7
Purity:  99.09%
Synonyms: LY3556050; CNTX-0290
Target:  

Somatostatin Receptor

Research Areas:  

Neurological Disease

Mazisotine (CNTX-0290) is an orally active, non-opioid somatostatin receptor 4 (SSTR4) agonist with an EC50 of 4.7 nM. Mazisotine exerts significant analgesic effects in various nociceptive (inflammatory, osteoarthritic) and neuropathic pain models. Mazisotine can be used for pain research .
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Cat. No.: HY-142699
CAS No.: 1638589-52-2
Target:  

Somatostatin Receptor

Research Areas:  

Inflammation/Immunology

SSTR4 agonist 2 is a potent agonist of somatostatin receptor subtype 4 (SSTR4). SSTR4 pathway inhibits nociceptive and inflammatory processes. SSTR4 agonist 2 has the potential for the research of medical disorders related to SSTR4 (extracted from patent WO2014184275A1, compound 107) .
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Cat. No.: HY-142701
CAS No.: 2747928-27-2
Target:  

Somatostatin Receptor

Research Areas:  

Neurological Disease

SSTR4 agonist 4 is a somatostatin receptor 4 (SSTR4) agonist. SSTR4 agonist 4 functionally activates SSTR4. SSTR4 agonist 4 has the potential for the research of pain .
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Cat. No.: HY-105172
CAS No.: 147159-51-1
Purity:  98.27%
Synonyms: CAP-232; TLN-232
Target:  

Somatostatin Receptor

Research Areas:  

Inflammation/Immunology Cancer

TT-232 (CAP-232), a somatostatin derivative, is a peptide SSTR1/SSTR4 agonist. TT-232 inhibits cancer cell proliferation and induces apoptosis. TT-232 is also a broad-spectrum anti-inflammatory and analgesic agent [4].
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Cat. No.: HY-172147
CAS No.: 2761347-44-6
Target:  

Somatostatin Receptor

Research Areas:  

Neurological Disease

SSTR4 agonist 5 (Compound 5) is the orally active agonist for somatostatin receptor 4 (SSTR4) with an EC50 of 0.228 nM. SSTR4 agonist 5 exhibits good stability in human/rat liver microsomes. SSTR4 agonist 5 inhibits mechanical hyperalgesia in rat models .
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Cat. No.: HY-142700
CAS No.: 2744188-34-7
Target:  

Somatostatin Receptor

Research Areas:  

Neurological Disease

SSTR4 agonist 3 is a potent agonist of SSTR4. SSTR4 is expressed at relatively high levels in the hippocampus and neocortex, memory and learning regions, and Alzheimer's disease pathology. SSTR4 agonists are potent in rodent models of pain associated with acute and chronic associated anti-peripheral nociceptive and anti-inflammatory activity. SSTR4 agonist 3 has the potential for the research of pain (extracted from patent WO2021233427A1, compound 14) .
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Cat. No.: HY-RS13829

SSTR4 Human Pre-designed siRNA Set A contains three designed siRNAs for SSTR4 gene (Human), as well as a negative control, a positive control, and a FAM-labeled negative control.

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Cat. No.: HY-RS13830

Sstr4 Mouse Pre-designed siRNA Set A contains three designed siRNAs for Sstr4 gene (Mouse), as well as a negative control, a positive control, and a FAM-labeled negative control.

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Cat. No.: HY-RS13831

Sstr4 Rat Pre-designed siRNA Set A contains three designed siRNAs for Sstr4 gene (Rat), as well as a negative control, a positive control, and a FAM-labeled negative control.

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Cat. No.: HY-W1117589
CAS No.: 2744188-17-6
Target:  

Somatostatin Receptor

Research Areas:  

Neurological Disease

SSTR4 agonist 6 (Compound 1) is a SSTR4 agonist. SSTR4 agonist 6 can be used for pain research .
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Cat. No.: HY-P3618
Cortistatin-29 is a neuropeptide. Cortistatin-29 alleviates neuropathic pain. Cortistatin-29 binds all somatostatin (SS) receptor subtypes with high affinity and shows IC50 values of 2.8 nM, 7.1 nM, 0.2 nM, 3.0 nM, 13.7 nM for SSTR1, SSTR2, SSTR3, SSTR4, SSTR5, respectively. Cortistatin-29 shows anti-fibrotic effects [4].
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Cat. No.: HY-P4555
CAS No.: 340821-13-8
Target:  

Somatostatin Receptor

Research Areas:  

Neurological Disease

(D-Phe5,Cys6,11,N-Me-D-Trp8)-Somatostatin-14 (5-12) amide (Compound 4) is a somatostatin analog with Kds of 0.61, 11.05, 23.5, 1200 and >1000 nM for SSTR5, SSTR3, SSTR2, SSTR1 and SSTR4, respectively .
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Cat. No.: HY-139347A
CAS No.: 2919211-45-1
Synonyms: LY3556050 tartrate; CNTX-0290 tartrate
Target:  

Somatostatin Receptor

Research Areas:  

Neurological Disease

Mazisotine (CNTX-0290) tartrate is an orally active, non-opioid somatostatin receptor 4 (SSTR4) agonist with an EC50 of 4.7 nM. Mazisotine tartrate exerts significant analgesic effects in various nociceptive (inflammatory, osteoarthritic) and neuropathic pain models. Mazisotine tartrate can be used for pain research .
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Cat. No.: HY-P2150
CAS No.: 1815618-17-7
Cortistatin-29 is a neuropeptide. Cortistatin-29 alleviates neuropathic pain. Cortistatin-29 binds all somatostatin (SS) receptor subtypes with high affinity and shows IC50 values of 2.8 nM, 7.1 nM, 0.2 nM, 3.0 nM, 13.7 nM for SSTR1, SSTR2, SSTR3, SSTR4, SSTR5, respectively. Cortistatin-29 shows anti-fibrotic effects [4].
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