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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
49 Results for "
arginine derivative
" in MedChemExpress (MCE) Product Catalog:
Products (49)
49 Results for "arginine derivative" in MCE Product Catalog:
2
2 Cited Publications
Synonyms: PAD2-IN-1 hydrochloride
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AFM32a (PAD2-IN-1) hydrochloride, a benzimidazole-based derivative, is a potent and selective protein arginine deiminase 2 (PAD2) inhibitor. AFM32a hydrochloride shows superior selectivity for PAD2 over PAD4 (95-fold) and PAD3 (79-fold) .
2
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Cardiovascular Disease Metabolic Disease Endocrinology Cancer
Mozavaptan (OPC-31260) is a benzazepine derivative and a potent, selective, competitive and orally active vasopressin V2 receptor antagonist with an IC50 of 14 nM. Mozavaptan shows ~85-fold selectivity for V2 receptor over V1 receptor (IC50 of 1.2 μM), and can antagonize the antidiuretic action of arginine vasopressin (AVP) in vivo. Mozavaptan has the potential for hyponatremia, syndrome of inappropriate antidiuretic hormone (SIADH), and congestive heart failure treatment .
2
2 Cited Publications
Synonyms: OPC-31260 hydrochloride
Target:
Research Areas:
Cardiovascular Disease Metabolic Disease Endocrinology Cancer
Mozavaptan hydrochloride (OPC-31260 hydrochloride) is a benzazepine derivative and a potent, selective, competitive and orally active vasopressin V2 receptor antagonist with an IC50 of 14 nM. Mozavaptan hydrochloride shows ~85-fold selectivity for V2 receptor over V1 receptor (IC50 of 1.2 μM), and can antagonize the antidiuretic action of arginine vasopressin (AVP) in vivo. Mozavaptan hydrochloride has the potential for hyponatremia, syndrome of inappropriate antidiuretic hormone (SIADH), and congestive heart failure treatment .
Cat. No.: HY-Y1636
CAS No.: 154445-77-9
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Cat. No.: HY-W099595
CAS No.: 60372-77-2
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Cat. No.: HY-W010698
CAS No.: 187618-60-6
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Cat. No.: HY-P10069
CAS No.: 2313534-24-4
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Cat. No.: HY-137002
CAS No.: 913733-27-4
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Cat. No.: HY-W008694
CAS No.: 2645-08-1
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Cat. No.: HY-W008389
CAS No.: 200124-22-7
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Cat. No.: HY-W008866
CAS No.: 401915-53-5
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Cat. No.: HY-W062304
CAS No.: 186698-61-3
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Cat. No.: HY-W040067
CAS No.: 2188-18-3
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Cat. No.: HY-W013305
CAS No.: 13726-76-6
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Cat. No.: HY-W010745
CAS No.: 83792-47-6
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Cat. No.: HY-W009211
CAS No.: 6382-93-0
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Cat. No.: HY-W089229
CAS No.: 776277-76-0
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Cat. No.: HY-W101935
CAS No.: 113712-06-4
Synonyms: N-Boc-D-arginine hydrochloride
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Cat. No.: HY-136557
CAS No.: 2095109-82-1
Synonyms: PAD2-IN-1
Target:
Research Areas:
AFM32a (PAD2-IN-1), a benzimidazole-based derivative, is a potent and selective protein arginine deiminase 2 (PAD2) inhibitor. AFM32a shows superior selectivity for PAD2 over PAD4 (95-fold) and PAD3 (79-fold) .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
