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7 Results for "
myosin I inhibitor
" in MedChemExpress (MCE) Product Catalog:
Products (7)
7 Results for "myosin I inhibitor" in MCE Product Catalog:
1
Phenamacril (JS399-19) inhibits activity of myosin I non-competitively with an IC50 of 360 nM through suppression of the ATPase activity, exhibits therefore an antifungal efficacy towards Fusarium species .
Cat. No.: HY-122200R
CAS No.: 39491-78-6
Synonyms: JS399-19 (Standard)
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Research Areas:
Phenamacril (Standard) is the analytical standard of Phenamacril. This product is intended for research and analytical applications. Phenamacril (JS399-19) inhibits activity of myosin I non-competitively with an IC50 of 360 nM through suppression of the ATPase activity, exhibits therefore an antifungal efficacy towards Fusarium species .
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Research Areas:
A-3 hydrochloride is a potent, cell-permeable, reversible, ATP-competitive non-selective antagonist of various kinases. It against PKA (Ki=4.3 µM), casein kinase II (Ki=5.1 µM) and myosin light chain kinase (MLCK) (Ki=7.4 µM). A-3 hydrochloride also inhibits PKC and casein kinase I with Ki values of 47 µM and 80 µM, respectively .
Cat. No.: HY-179120
CAS No.: 3095661-21-2
ZJS178 is a novel inhibitor of myosin I. ZJS178 is a fungicide that has inhibitory activity against Fusarium graminearum and can reduce DON toxin synthesis. ZJS178 can be used for research on plant diseases such as wheat scab .
Cat. No.: HY-189346
Myosin I-IN-1 is an Antifungal agent and Myosin I inhibitor with a Kd of 0.14 μM for FgMyoI. Myosin I-IN-1 inhibits mycelial growth, sporulation, spore germination, and Deoxynivalenol (HY-N6684) biosynthesis. Myosin I-IN-1 disrupts cell wall and cell membrane integrity and induces hyphal morphological changes. Myosin I-IN-1 exhibits broad-spectrum antifungal activity against plant pathogenic fungi. Myosin I-IN-1 shows protective efficacy against Fusarium head blight in wheat and maize. Myosin I-IN-1 can be used for research on Fusarium head blight .
Cat. No.: HY-189456
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Antifungal agent 183 is a Myosin I inhibitor (Kd = 0.37 μM) that binds to the conserved phenamacril-binding pocket in the motor domain of Botrytis cinerea myosin I, inhibits Actin-dependent ATPase activity, and blocks the ATPase cycle, thereby disrupting hyphal tip morphogenesis and inhibiting hyphal and colony growth. Antifungal agent 183 can be used for research on gray mold .
Cat. No.: HY-W718178
CAS No.: 152-84-1
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Protocols
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