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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
9 Results for "
willardiine
" in MedChemExpress (MCE) Product Catalog:
Products (9)
9 Results for "willardiine" in MCE Product Catalog:
Synonyms: (-)-willardiine
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Research Areas:
(S)-Willardiine ((-)-Willardiine) is a subtype-selective glutamate receptor agonist and the active isomer of Willardiine. Willardiine binds to and activates hGluR1, hGluR2, hGluR4 and hGluR5, with Ki values of 3.6 nM and 0.24 nM for hGluR4 and hGluR5, respectively. (S)-Willardiine is used to investigate the distribution and physiological functions of glutamate receptor subunits in the central nervous system .
Cat. No.: HY-107606A
Purity: 97.48%
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UBP301 hydrochloride is a potent and selective antagonist of kainate receptor with IC50 and KD of 164 μM and 5.94 μM, respectively. UBP301 hydrochloride has ～30-fold selectivity of kainate receptor over AMPA receptor. UBP301 hydrochloride is the derivative of willardiine .
Cat. No.: HY-19432
CAS No.: 544697-47-4
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UBP-282 is a potent, selective and competitive AMPA and kainate receptor antagonist. UBP-282 inhibits the fast component of the dorsal root-evoked ventral root potential (fDR-VRP) with an IC50 value of 10.3 μM. UBP-282 antagonizes kainate-induced depolarisations of dorsal roots with a pA2 value of 4.96 .
Cat. No.: HY-W922811
CAS No.: 19772-76-0
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DL-Willardiine is an AMPA antagonist with an IC50 of 2 μM. DL-Willardiine can be utilized in psychotropic cccccc research .
Cat. No.: HY-CE01781
Synonyms: Fluoro-willardiine-coenzyme A
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Fluoro-willardiine-CoA (Fluoro-willardiine-coenzyme A) is a coenzyme A derivative .
Cat. No.: HY-CE01837
Synonyms: Iodo-willardiine-coenzyme A
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Iodo-willardiine-CoA (Iodo-willardiine-coenzyme A) is a coenzyme A derivative .
Cat. No.: HY-107606
CAS No.: 569371-10-4
Target:
Research Areas:
UBP301 is a potent and selective antagonist of kainate receptor with IC50 and KD of 164 μM and 5.94 μM, respectively. UBP301 has ∼30-fold selectivity of kainate receptor over AMPA receptor. UBP301 is the derivative of willardiine .
Cat. No.: HY-CE01903
Synonyms: willardiine-coenzyme A
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Willardiine-CoA (Willardiine-coenzyme A) is a coenzyme A derivative .
Cat. No.: HY-CE01235
Synonyms: Bromo-willardiine-coenzyme A
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Research Areas:
Bromo-willardiine-CoA (Bromo-willardiine-coenzyme A) is a coenzyme A derivative .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
