1. Membrane Transporter/Ion Channel
    Neuronal Signaling
  2. GABA Receptor
  3. THIP

THIP (Synonyms: Gaboxadol)

Cat. No.: HY-10232
Handling Instructions

THIP (Gaboxadol) is a selective δ-aminobutyric acid type A receptor (δ-GABAAR) agonist, functionally selective GABAAR ligand, exhibits agonism at α4β1δ, α4β3δ and weak antagonism at αβγ and α4β2δ GABAARs.

For research use only. We do not sell to patients.

THIP Chemical Structure

THIP Chemical Structure

CAS No. : 64603-91-4

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Description

THIP (Gaboxadol) is a selective δ-aminobutyric acid type A receptor (δ-GABAAR) agonist, functionally selective GABAAR ligand, exhibits agonism at α4β1δ, α4β3δ and weak antagonism at αβγ and α4β2δ GABAARs[1].

IC50 & Target

α4β3δ GABAAR

13 μM (EC50)

Molecular Weight

140.14

Formula

C₆H₈N₂O₂

CAS No.

64603-91-4

SMILES

O=C1C2=C(CNCC2)ON1

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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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THIP
Cat. No.:
HY-10232
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