1. PROTAC
  2. E3 Ligase Ligand-Linker Conjugate
  3. (S,R,S)-AHPC-PEG4-NH2

(S,R,S)-AHPC-PEG4-NH2 (Synonyms: VH032-PEG4-NH2; VHL Ligand-Linker Conjugates 4 ; E3 ligase Ligand-Linker Conjugates 7 Free Base)

Cat. No.: HY-103604A Purity: 98.26%
Handling Instructions

(S,R,S)-AHPC-PEG4-NH2 is a synthesized E3 ligase ligand-linker conjugate that incorporates the (S,R,S)-AHPC based VHL ligand and 4-unit PEG linker used in PROTAC technology.

For research use only. We do not sell to patients.

(S,R,S)-AHPC-PEG4-NH2 Chemical Structure

(S,R,S)-AHPC-PEG4-NH2 Chemical Structure

CAS No. : 2010159-57-4

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 605 In-stock
Estimated Time of Arrival: December 31
100 mg USD 550 Get quote
500 mg USD 1950 Get quote
1 g USD 3350 Get quote
2 g USD 4900 Get quote
5 g   Get quote  
10 g   Get quote  

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Description

(S,R,S)-AHPC-PEG4-NH2 is a synthesized E3 ligase ligand-linker conjugate that incorporates the (S,R,S)-AHPC based VHL ligand and 4-unit PEG linker used in PROTAC technology.

IC50 & Target[1]

VHL

 

In Vitro

E3 ligase Ligand-Linker Conjugates 7 Free Base, extracted from patent US20170008904A1, can be used in the synthesis of compound A1895 in example 3[1].

Molecular Weight

663.83

Formula

C₃₂H₄₉N₅O₈S

CAS No.

2010159-57-4

SMILES

O=C(N[[email protected]@H](C(C)(C)C)C(N(C[[email protected]](O)C1)[[email protected]@H]1C(NCC2=CC=C(C(SC=N3)=C3C)C=C2)=O)=O)COCCOCCOCCOCCN

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
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Keywords:

(S,R,S)-AHPC-PEG4-NH2VH032-PEG4-NH2VHL Ligand-Linker Conjugates 4 E3 ligase Ligand-Linker Conjugates 7E3 Ligase Ligand-Linker ConjugateInhibitorinhibitorinhibit

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Product name:
(S,R,S)-AHPC-PEG4-NH2
Cat. No.:
HY-103604A
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