1. GPCR/G Protein
  2. Angiotensin Receptor
  3. SL910102

SL910102 

Cat. No.: HY-100292
Handling Instructions

SL910102 is a nonpeptide angiotensin AT1 receptor antagonist.

For research use only. We do not sell to patients.

SL910102 Chemical Structure

SL910102 Chemical Structure

CAS No. : 144756-71-8

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Description

SL910102 is a nonpeptide angiotensin AT1 receptor antagonist.

IC50 & Target

Angiotensin AT1 receptor[1]

In Vitro

SL910102 (SL 91.0102-90 DL) is a unlabelled nonpeptide AT1-antagonist, which is tested for its ability to compete with [125J](Sar1-Ile8)-angiotensin II for specific AT1-receptor sites in rat lung homogenate[1].

Molecular Weight

490.60

Formula

C₃₀H₃₀N₆O

CAS No.

144756-71-8

SMILES

O=C1N=C(CCC2=CC=CC=C2)NC(CCCC)=C1CC3=CC=C(C4=CC=CC=C4C5=NN=NN5)C=C3

Shipping

Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
Kinase Assay
[1]

For saturation as well as displacement studies, rat lung homogenate is incubated in either Hepes-buffer or blank human or rat plasma yielding 50 μg protein per well in a total assay volume of 300 μL. To ensure equilibrium conditions (see binding kinetics), the samples are maintained for 60 min at 25°C under continuous rotation. All experiments are carried out in duplicate, and the results are confirmed with n=3-5 replicates over the following days[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

References
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