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  2. Thyroid Hormone Receptor
  3. Taltirelin

Taltirelin (Synonyms: TA-0910)

Cat. No.: HY-B0596 Purity: >98.0%
Handling Instructions

Taltirelin (TA0910) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release).

For research use only. We do not sell to patients.

Taltirelin Chemical Structure

Taltirelin Chemical Structure

CAS No. : 103300-74-9

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 66 In-stock
Estimated Time of Arrival: December 31
5 mg USD 60 In-stock
Estimated Time of Arrival: December 31
10 mg USD 96 In-stock
Estimated Time of Arrival: December 31
50 mg USD 384 In-stock
Estimated Time of Arrival: December 31
100 mg USD 696 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

Other Forms of Taltirelin:

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Description

Taltirelin (TA0910) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release)[1].

IC50 & Target

IC50: 910 nM (Thyrotropin-releasing hormone receptor)[1]

Molecular Weight

405.41

Formula

C₁₇H₂₃N₇O₅

CAS No.

103300-74-9

SMILES

O=C(N(CCC1)[[email protected]@H]1C(N)=O)[[email protected]@H](NC([[email protected]@H](NC2=O)CC(N2C)=O)=O)CC3=CN=CN3

Shipping

Room temperature in continental US; may vary elsewhere

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : ≥ 32 mg/mL (78.93 mM)

*"≥" means soluble, but saturation unknown.

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Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.4666 mL 12.3332 mL 24.6664 mL
5 mM 0.4933 mL 2.4666 mL 4.9333 mL
10 mM 0.2467 mL 1.2333 mL 2.4666 mL
*Please refer to the solubility information to select the appropriate solvent.
References
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Taltirelin
Cat. No.:
HY-B0596
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