1. Signaling Pathways
  2. Cell Cycle/DNA Damage
    Cytoskeleton
  3. PAK
  4. PAK Inhibitors

PAK Inhibitors

PAK1

PAK2

PAK3

PAK4

PAK5

PAK6

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

PAK Inhibitors & Activators
Product Name PAK1 PAK2 PAK3 PAK4 PAK5 PAK6 Purity
Fingolimod hydrochloride
PAK1
          99.95%
5-Aminosalicylic Acid
PAK1
          ≥98.0%
Fingolimod
PAK1
          99.56%
PF-3758309
PAK1, Ki: 13.7 nM
PAK2, IC50: 190 nM
PAK3, IC50: 99 nM
PAK4, Ki: 18.7 nM
PAK4, Kd: 2.7 nM
PAK5, Ki: 18.1 nM
PAK6, Ki: 17.1 nM
99.84%
IPA-3
PAK1, IC50: 2.5 μM
          99.43%
FRAX597
PAK1, IC50: 8 nM
PAK2, IC50: 13 nM
PAK3, IC50: 19 nM
      99.79%
FRAX486
PAK1, IC50: 14 nM
PAK2, IC50: 33 nM
PAK3, IC50: 39 nM
      98.01%
G-5555
PAK1, Ki: 3.7 nM
PAK2, Ki: 11 nM
        99.29%
Padnarsertib      
PAK4, IC50: 100 nM
    99.86%
LCH-7749944      
PAK4, IC50: 14.93 μM
    99.36%
G-5555 hydrochloride
PAK1, Ki: 3.7 nM
PAK2, Ki: 11 nM
        98.78%
AZ13705339
PAK1, Kd: 0.28 nM
PAK1, IC50: 0.33 nM
pPAK1, IC50: 59 nM
PAK2, Kd: 0.32 nM
        98.90%
AZ13705339 hemihydrate
PAK1, Kd: 0.28 nM
PAK1, IC50: 0.33 nM
pPAK1, IC50: 59 nM
PAK2, Kd: 0.32 nM
        99.77%
PAK4-IN-2    
PAK3, IC50: 2.7 nM
      99.78%
PAK1-IN-1
PAK1, IC50: 9.8 nM
   
PAK4, IC50: >10 μM
   
PF-3758309 hydrochloride
PAK1, Ki: 13.7 nM
PAK2, IC50: 190 nM
PAK3, IC50: 99 nM
PAK4, Ki: 18.7 nM
PAK4, Kd: 2.7 nM
PAK5, Ki: 18.1 nM
PAK6, Ki: 17.1 nM
PF-3758309 dihydrochloride
PAK1, Ki: 13.7 nM
PAK2, IC50: 190 nM
PAK3, IC50: 99 nM
PAK4, Ki: 18.7 nM
PAK4, Kd: 2.7 nM
PAK5, Ki: 18.1 nM
PAK6, Ki: 17.1 nM
G-9791
PAK1, Ki: 0.95 nM
PAK2, Ki: 2.0 nM
       
NVS-PAK1-C
PAK1, Kd: 0.007 μM
PAK1, IC50: 5 nM
PAK2, Kd: 0.4 μM
PAK2, IC50: 270 nM
        ≥99.0%
Mesalamine impurity P
PAK1
         
PAK4-IN-1      
PAK4
   
ZINC194100678
PAK1, IC50: 8.37 μM
         
ZMF-10
PAK1, IC50: 174 nM
PAK2, IC50: 1.038 μM
PAK3, IC50: 1.372 μM