1. Signaling Pathways
  2. Protein Tyrosine Kinase/RTK
  3. PDGFR
  4. PDGFR Inhibitors

PDGFR Inhibitors

PDGFR

PDGFRβ

PDGFRα

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

PDGFR Inhibitors
Product Name PDGFR PDGFRβ PDGFRα Purity
Lenvatinib  
PDGFRβ, IC50: 39 nM
PDGFRα, IC50: 51 nM
99.84%
Sunitinib  
PDGFRβ, IC50: 2 nM
  98.96%
Regorafenib  
PDGFRβ, IC50: 22 nM
  99.65%
Nintedanib  
PDGFRβ, IC50: 65 nM
PDGFRα, IC50: 59 nM
99.82%
Ponatinib hydrochloride    
PDGFRα, IC50: 1.1 nM
99.26%
Tovetumab    
PDGFRα
99.49%
Regorafenib mesylate  
PDGFRβ, IC50: 22 ± 3 nM
 
Ponatinib    
PDGFRα, IC50: 1.1 nM
99.43%
Axitinib  
PDGFRβ, IC50: 1.6 nM
  99.94%
Pazopanib  
PDGFRβ, IC50: 84 nM
  99.77%
Crenolanib  
PDGFRβ, Kd: 3.2 nM
PDGFRα, Kd: 2.1 nM
99.72%
SU 5402  
PDGFRβ, IC50: 510 nM
  99.38%
Linifanib  
PDGFRβ, IC50: 66 nM
  99.72%
Sunitinib Malate  
PDGFRβ, IC50: 2 nM
  99.91%
Nintedanib esylate  
PDGFRβ, IC50: 65 nM
PDGFRα, IC50: 59 nM
99.94%
Ripretinib    
PDGFRA
99.33%
Dovitinib  
PDGFRβ, IC50: 27 nM
PDGFRα, IC50: 210 nM
99.94%
Cediranib  
PDGFRβ, IC50: 5 nM
PDGFRα, IC50: 36 nM
99.58%
Lenvatinib mesylate  
PDGFRβ, IC50: 39 nM
PDGFRα, IC50: 51 nM
99.86%
CP-673451  
PDGFRβ, IC50: 1 nM
PDGFRα, IC50: 10 nM
99.65%
Pazopanib Hydrochloride  
PDGFRβ, IC50: 84 nM
  99.88%
ENMD-2076    
PDGFRα, IC50: 56.4 nM
99.12%
Telatinib    
PDGFRα, IC50: 15 nM
99.60%
CHIR-124
PDGFR, IC50: 6.6 nM
    98.57%
Amuvatinib    
PDGFRαV561D, IC50: 40 nM
PDGFRαD842V, IC50: 81 nM
98.07%
PP121
PDGFR, IC50: 2 nM
    99.08%
Regorafenib Hydrochloride  
PDGFRβ, IC50: 22 nM
  99.58%
SU14813  
PDGFRβ, IC50: 4 nM
  99.63%
Orantinib  
PDGFRβ, Ki: 8 nM
  99.13%
Tandutinib
PDGFR, IC50: 0.2 μM
    99.48%
TAK-593  
PDGFRβ, IC50: 13 nM
PDGFRα, IC50: 4.3 nM
PDGFRαV561D, IC50: 1 nM
99.62%
Flumatinib mesylate  
PDGFRβ, IC50: 307.6 nM
  99.87%
Regorafenib monohydrate  
PDGFRβ, IC50: 22 nM
  99.96%
Dovitinib lactate  
PDGFRβ, IC50: 210 nM
PDGFRα, IC50: 27 nM
99.62%
Cediranib maleate  
PDGFRβ, IC50: 5 nM
PDGFRα, IC50: 36 nM
99.84%
Chiauranib  
PDGFRβ, IC50: 93 nM
PDGFRα, IC50: 1 nM
99.28%
Tyrphostin AG1296  
PDGFRβ
PDGFRα
99.25%
Ilorasertib hydrochloride  
PDGFRβ, IC50: 13 nM
PDGFRα, IC50: 11 nM
99.67%
TG 100801  
PDGFRβ, IC50: 13 nM
  98.60%
AZD2932  
PDGFRβ, IC50: 4 nM
  ≥98.0%
Toceranib phosphate  
PDGFRβ, Ki: 5 nM
  98.02%
JNJ-10198409  
PDGFRβ, IC50: 4.2 nM
PDGFRα, IC50: 45 nM
≥99.0%
Tyrosine kinase-IN-1    
PDGFRα, IC50: 4 nM
99.34%
PP58
PDGFR
    99.48%
JI-101  
PDGFRβ
  99.43%
Toceranib  
PDGFRβ, Ki: 5 nM
 
Telatinib mesylate    
PDGFRα, IC50: 15 nM
99.46%
(Z)-Orantinib  
PDGFRβ, IC50: 0.008 μM
  99.02%
PD-161570
PDGFR, IC50: 310 nM
PDGFRβ, IC50: 262 nM
  99.04%
SU4312
PDGFR
    98.19%
ENMD-2076 Tartrate    
PDGFRα, IC50: 56.4 nM
98.87%
AC710  
PDGFRβ, Kd: 1 nM
PDGFRα, Kd: 1.3 nM
99.89%
Famitinib  
PDGFRβ, IC50: 6.6 nM
  98.09%
SU16f
PDGFR2, IC50: 140 nM
PDGFR1, IC50: 2.29 μM
PDGFRβ, IC50: 10 nM
  ≥99.0%
Methylnissolin
PDGFR, IC50: 10 μM
    99.64%
Hypothemycin  
PDGFRβ, Ki: 900 nM
PDGFRα, Ki: 1.5 μM
≥98.0%
GZD856 formic  
PDGFRβ, IC50: 136.6 nM
PDGFRα, IC50: 68.6 nM
98.06%
Tyrphostin AG1433  
PDGFRβ, IC50: 5 μM
  99.20%
Tandutinib hydrochloride
PDGFR, IC50: 0.2 μM
    99.78%
PDGFRα kinase inhibitor 1  
PDGFRβ, IC50: 6115 nM
PDGFRα, IC50: 132 nM
99.78%
Zeteletinib
PDGFR2
    99.06%
KG5  
PDGFRβ, Kd: 520 nM
PDGFRα, Kd: 300 nM
99.79%
SU14813 maleate  
PDGFRβ, IC50: 4 nM
  99.04%
NVP-ACC789  
PDGFR-β, IC50: 1.4 μM
  99.94%
Sunitinib-d10  
PDGFRβ, IC50: 2 nM
  99.89%
Ponatinib-d8    
PDGFRα, IC50: 1.1 nM
98.44%
TG 100572  
PDGFRβ, IC50: 13 nM
 
Ilorasertib  
PDGFRβ, IC50: 13 nM
PDGFRα, IC50: 11 nM
≥98.0%
Dovitinib lactate hydrate  
PDGFRβ, IC50: 210 nM
PDGFRα, IC50: 27 nM
GZD856  
PDGFRβ, IC50: 136.6 nM
PDGFRα, IC50: 68.6 nM
Zeteletinib hemiadipate
PDGFR2
   
Famitinib malate  
PDGFRβ, IC50: 6.6 nM
 
Amuvatinib hydrochloride    
PDGFRαV561D, IC50: 40 nM
PDGFRαD842V, IC50: 81 nM
Multi-kinase-IN-1    
PDGFRα, IC50: 0.384 μM
PD-089828  
PDGFR-β, IC50: 1.76 μM
PDGFR-β, Ki: 2.38 μM
 
Multi-kinase inhibitor 1
PDGFR
   
AG 370
PDGFR, IC50: 20 μM
   
Multi-kinase-IN-2  
PDGFRβ, IC50: 9.9 ± 0.7 nM
PDGFRα, IC50: 7.0 ± 0.1 nM
Multi-kinase-IN-3  
PDGFRβ, IC50: 55 ± 2.6 nM
 
HG-7-85-01    
PDGFRα, IC50: 440 nM
IHMT-TRK-284  
PDGFRβ, IC50: 95.7 nM
PDGFRα, IC50: 24.2 nM
Henatinib  
PDGFRβ
PDGFRα
TG 100801 Hydrochloride  
PDGFRβ, IC50: 13 nM
 
AC710 Mesylate  
PDGFRβ, Kd: 1 nM
PDGFRα, Kd: 1.3 nM