ROR Inhibitors

RORγ

RORα

RORβ

ROR Inhibitors, Agonists, Antagonists, Activators, Modulators & Ligands

Product Name	RORγ	RORα	RORβ	Purity
RORγ-IN-3	ROR-γ, EC₅₀: 84 nM
Lithocholic acid 3-sulfate disodium	RORγt, Kd: 1.7×10<sup			99.93%
Allolithocholic acid	RORγt, IC₅₀: 3.4 μM			99.69%
XY018	ROR-γ, IC₅₀: 0.19 μM (in 293 T cells)	ROR-α, IC₅₀: 7.57 μM (in 293 T cells)		99.68%
Zymostenol	RORγ, EC₅₀: 1 μM			99.33%
GNE-6468	ROR-γ, EC₅₀: 2 nM			98.02%
F44-A13	RORγ
Izumerogant	RORγ, IC₅₀: 10 nM			99.95%
JNJ-61803534	RORγt			99.84%
(±)-ML 209	RORγ, IC₅₀: 1.1 μM			98.14%
7ß,27-Dihydroxycholesterol	RORγt, Ki: 120 nM			99.5%
RORγt inverse agonist 13	ROR-γ, IC₅₀: 63.8 nM			98.13%
SR1555	RORγ, IC₅₀: 1 μM			99.69%
GNE-3500	ROR-γ, EC₅₀: 12 nM			98.90%
Vimirogant hydrochloride	RORγt, Ki: 3.5 nM RORγt, IC₅₀: 17 nM			98.39%
RORγt Inverse agonist 10	RORγt, IC₅₀: 51 nM			99.13%
S18-000003	RORγt, IC₅₀: <30 nM			99.31%
Hexyl 4-hydroxybenzoate	RORγt, EC₅₀: 144 nM			99.83%
BMS-986251	RORγt, EC₅₀: 12 nM	RORα, EC₅₀: >10 μM	RORβ, EC₅₀: >10 μM
W6134	RORγ, IC₅₀: 0.21 μM			99.90%
A-9758	RORγt, IC₅₀: 5 nM
SHR168442	ROR-γ
RORγt inverse agonist 35	RORγt, IC₅₀: 1.51 μM
RORγt modulator 5	RORγt, Ki: <100 nM
RORγt modulator 4	RORγt
RORγt inhibitor 4	RORγt
RORγt inverse agonist 33	RORγt, IC₅₀: 21 nM
XY039	RORγ, IC₅₀: 0.55 μM
RORγ agonist 2	RORγ, EC₅₀: 0.03 μM	RORα, EC₅₀: >3 μM
RORγt inverse agonist 34	RORγt, IC₅₀: 0.094 μM
RORγt inverse agonist 37	RORγt, IC₅₀: 10.8 nM
RORγt inverse agonist 32	RORγt
BMS-336	RORγ
RORγt inverse agonist 29	RORγt, IC₅₀: 21 nM
Gala-SR		RORα
CD12681	RORγ
RORγ-IN-2	RORγ, Ki: 16.6 nM
RORγt inverse agonist 36	RORγt
RORγ-IN-4	RORγ, EC₅₀: 0.014 μM
RORγt inverse agonist 30	RORγt, IC₅₀: 46 nM
CID 7309015	ROR-γ
SR-1903	RORγ, IC₅₀: ~100 nM
Vimirogant	RORγt, Ki: 3.5 nM RORγt, IC₅₀: 17 nM

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