1. Signaling Pathways
  2. Stem Cell/Wnt
  3. YAP
  4. YAP Inhibitors

YAP Inhibitors

YAP/TAZ

YAP/TAZ-TEAD

TEAD

YAP1

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YAP Inhibitors, Antagonists, Activators, Modulators, Degraders & Ligands
Product Name YAP/TAZ YAP/TAZ-TEAD TEAD YAP1 Purity
Verteporfin  
YAP/TAZ-TEAD
    99.58%
KG-FP-003    
TEAD1, DC50: 6 nM
TEAD2, DC50: 68 nM
TEAD3, DC50: 12 nM
 
TEAD ligand 2    
TEAD1
 
IAG933  
YAP/TAZ-TEAD
    99.47%
GNE-7883  
YAP/TAZ-TEAD
    99.54%
ML-7 hydrochloride
YAP/TAZ
      99.88%
GA-017
YAP/TAZ
      98.95%
Thiostrepton  
YAP/TAZ-TEAD
    99.80%
Ki16425
YAP/TAZ
      98.88%
VT3989
YAP/TAZ
      99.61%
TED-347  
YAP/TAZ-TEAD
    99.13%
YAP/TAZ inhibitor-1
YAP/TAZ
      99.72%
MYF-03-69    
TEAD1, IC50: 385 nM
TEAD2, IC50: 143 nM
TEAD3, IC50: 558 nM
  98.11%
SWTX-143  
YAP/TAZ-TEAD
    99.81%
Super-TDU  
YAP/TAZ-TEAD
    99.65%
YAP-TEAD-IN-1  
YAP/TAZ-TEAD
    99.68%
YAP/TAZ inhibitor-2  
YAP/TAZ-TEAD
    99.81%
YAP-TEAD-IN-1 TFA
YAP/TAZ
      99.99%
TEAD1/3/4-IN-1  
YAP/TAZ-TEAD, EC50: 2 nM
    99.04%
PROTAC TEAD degrader-1    
TEAD2, DC50: 32.7 nM
  99.82%
MSC-4106  
YAP/TAZ-TEAD
    99.87%
MYF-01-37  
YAP/TAZ-TEAD
    99.34%
TEAD-IN-1    
TEAD
  99.43%
TD034      
YAP1
99.77%
TEAD-IN-8  
YAP/TAZ-TEAD
    99.84%
YTP-17  
YAP/TAZ-TEAD
    98.04%
(7S)-BAY-593  
YAP/TAZ-TEAD
    99.61%
Super-TDU (1-31)  
YAP/TAZ-TEAD
   
Super-TDU (1-31) TFA  
YAP/TAZ-TEAD
    99.27%
TEAD ligand 1    
TEAD2
 
TEAD ligand 4    
TEAD1
 
M3686    
TEAD1, IC50: 51 nM
 
OPN-9652    
TEAD, IC50: 0.005 μM
  98.84%
PROTAC TEAD1/IAP degrader-1    
TEAD1, DC50: 14 nM
 
TEAD-IN-21    
TEAD, IC50: 3 nM
 
TEAD ligand 5    
TEAD
 
LC-TEAD01    
TEAD, IC50: 116 nM
TEAD, Ki: 0.132 μM
 
OPN-9643    
TEAD, IC50: 15 nM
 
EA-C15    
TEAD, IC50: 0.34 μM
 
YAP/TAZ-TEAD-IN-2  
YAP/TAZ-TEAD
   
VT102    
TEAD1, IC50: 391 nM
 
TEAD-IN-23    
TEAD, IC50: 0.01 μM
 
Verteporfin (Standard)  
YAP/TAZ-TEAD
   
PROTAC TEAD1/IAP degrader-3    
TEAD1
 
N-Acetylgalactosaminyltransferase 12      
YAP1
MY-1576
YAP/TAZ
     
Super-TDU TFA  
YAP/TAZ-TEAD
   
TEAD ligand 6    
TEAD
 
PROTAC TEAD degrader-2  
YAP/TAZ-TEAD, IC50: 1.8 nM
TEAD1, DC50: 0.6 nM
 
CV-4-26  
YAP/TAZ-TEAD
   
YAP/TAZ-TEAD-IN-3  
YAP/TAZ-TEAD, IC50: 1.8 nM
   
pan-TEAD-IN-1    
TEAD
 
LATS1/2-IN-1      
YAP1
VT101    
TEAD, IC50: 454 nM
 
DC-TEAD3in03    
TEAD3, IC50: 0.16 μM
 
PROTAC TEAD/IAP degrader-1    
TEAD1
 
TEAD-IN-6  
YAP/TAZ-TEAD
   
TEAD-IN-9    
TEAD1, IC50: 0.29 μM
 
PROTAC TEAD1/IAP degrader-2    
TEAD1, DC50: 170 nM
 
TEAD ligand-Linker Conjugate 2    
TEAD
 
TEAD-IN-24    
TEAD
 
YAP/TAZ inhibitor-4
YAP/TAZ
YAP/TAZ-TEAD
   
TEAD ligand-Linker Conjugate 3    
TEAD1
 
TEAD ligand 3    
TEAD