Drug Derivative
Drug derivative
Drug derivatives are derived from parent compounds. They replace or add atoms and groups through chemical reactions to optimize the various properties of the parent compound and reduce side effects. The application of drug derivatives provides a diverse compound library for drug research and development and accelerates the discovery of new drugs. For example, urea derivatives Glibenclamide can prolong the blood sugar-lowering effect of anti-diabetic drugs.
References:
- [1]. Vardanyan RS, et al. Fentanyl-related compounds and derivatives: current status and future prospects for pharmaceutical applications. Future Med Chem. 2014 Mar;6(4):385-412.x
- [2]. Ghosh AK, et al. Urea Derivatives in Modern Drug Discovery and Medicinal Chemistry. J Med Chem. 2020 Mar 26;63(6):2751-2788.x
All Product Categories
-
Drug Derivative Inhibitors
(12)
View all products
-
Drug Derivative Agonist
(1)
View all products
-
Drug Derivative Activator
(1)
View all products
-
Drug Derivative Chemical
(1)
View all products
-
Drug Derivative Inducer
(1)
View all products
-
Drug Derivative Controls
(38)
View all products
-
Drug Derivative Substrate
(1)
View all products
-
Drug Derivative Related Products (4062)
Related Products (4062)
-
5-Deazaisofolic acid
0 ImagesCat. No.: HY-125420CAS No.: 130327-67-25-Deazaisofolic acid is an isofolate analogue with antitumor activity. 5-Deazaisofolic acid can be utilized in cancer research.
-
25,26,27-Trinor-3α-hydroxycycloartan-24-oic acid
0 ImagesCat. No.: HY-N17042CAS No.: 1300747-31-225,26,27-Trinor-3α-hydroxycycloartan-24-oic acid is a natural triterpene.
-
7,4'-Di-O-methylaromadendrin
0 ImagesCat. No.: HY-N17155CAS No.: 41515-76-87,4'-Di-O-methylaromadendrin is a natural flavonoid.
-
3,3',5'-Trihydroxy-4-methoxybibenzyl
0 ImagesCat. No.: HY-W1053643CAS No.: 60640-97-33,3',5'-Trihydroxy-4-methoxybibenzyl is a dihydrostilbene derivative that can be found in the leaves of Glycyrrhiza glabra.
-
Fenyramidol
0 ImagesCat. No.: HY-W748379CAS No.: 553-69-5Synonyms: (±)-PhenyramidolFenyramidol is an Aminopyridine derivative. Fenyramidol can be used as a moderately potent, non-narcotic muscle relaxant with concomitant analgesic activity.
-
TL-310
0 ImagesCat. No.: HY-119214CAS No.: 352697-38-2TL-310 is a novel, orally active Taxane analogue. TL-310 can be used in the research of solid tumors.
-
IDN-5404
0 ImagesCat. No.: HY-105943CAS No.: 361169-05-3
-
β-Carotene 5,6-epoxide
0 ImagesCat. No.: HY-W750682CAS No.: 1923-89-3β-Carotene 5,6-epoxide, a carotenoid, is a degradation product of β-carotene. β-Carotene 5,6-epoxide can be found in isolated chloroplasts. Carotenoids are important biological active, and may regulate cellular differentiation, growth control, photooxidative protection, cell membrane stability, photosynthesis, vision process and nutrition.
-
R-4066
0 ImagesCat. No.: HY-171234CAS No.: 66194-36-3R-4066 is an agent which is an analogue of the opioid analgesic Methadone. R-4066 is a highly potent, long-acting analgesic.
-
(-)-δ-Cadinene
0 ImagesCat. No.: HY-N18244CAS No.: 13061-82-0(-)-δ-Cadinene is a sesquiterpene found in the red seaweed Laurencia microcladia (Rhodophyta).
-
Descarbamylnovobiocin
0 ImagesCat. No.: HY-137806CAS No.: 75057-97-5Descarbamylnovobiocin is a derivative of Novobiocin (HY-B0425).
-
Anticancer agent 283
0 ImagesCat. No.: HY-179298Anticancer agent 283 (Compound 25) is a Forsyshiyanine A derivative. Anticancer agent 283 shows anticancer activity against pancreatic cancer.
-
1(R)-Tetrahydrocannabidiphorol
0 ImagesCat. No.: HY-1728481(R)-Tetrahydrocannabidiphorol is a drug analogue and can be used for the research of neurological disease.
-
Epimedonin G
0 ImagesCat. No.: HY-N9673CAS No.: 2222285-80-3Epimedonin G is a 2-phenoxychromone compound found in Epimedium brevicornum. Epimedonin G can be used for the research of cancer.
-
WAY-313165
0 ImagesWAY-313165 is an active molecule.
-
Timosaponin G
0 ImagesCat. No.: HY-N18255CAS No.: 195304-82-6Timosaponin G is a steroidal saponin found in the rhizomes of Anemarrhena asphodeloides.
-
KP-10614
0 ImagesCat. No.: HY-105514CAS No.: 130273-99-3KP-10614 is a potent, orally active platelet aggregation inhibitor. KP-10614 inhibits platelet aggregation induced by ADP with IC50 of 1 nM. KP-10614 causes dose-dependent inhibition of ex vivo platelet aggregation in rats. KP-10614 shows antithrombotic effects in various thrombosis models. KP-10614 can be used for thrombotic diseases research.
-
5-Hydroxy-3′,4′,7,8-tetramethoxyflavone
0 ImagesCat. No.: HY-N17979CAS No.: 13003-74-25-Hydroxy-3′,4′,7,8-tetramethoxyflavone is a flavone found in the whole plant of Peperomia sui. 5-Hydroxy-3′,4′,7,8-tetramethoxyflavone shows no activity against cancer cell lines in vitro.
