Tie Inhibitors

Tie1

Tie2

Tie Inhibitors & Activators

Product Name	Tie1	Tie2	Purity
Regorafenib		Tie2, IC₅₀: 311 ± 46 nM	99.93%
Regorafenib monohydrate		Tie2, IC₅₀: 311 ± 46 nM	99.94%
BAY-826		Tie2, Kd: 1.6 nM	99.94%
6-Hydroxy-2,2′,4,4′-tetrabromodiphenyl ether		Tie2
TP-S1-68		Tie2, IC₅₀: 3.65 μM
Tie2 kinase inhibitor 1		Tie2, IC₅₀: 250 nM	99.80%
NVP-BAW2881		Tie2, IC₅₀: 650 nM	98.54%
TIE-2/VEGFR-2 kinase-IN-2		Tie2, pIC₅₀: 8.56 nM	99.81%
Gersizangitide		Tie2
Tie2 kinase inhibitor 2		Tie2, IC₅₀: 1 μM Tie2, IC₅₀: 1.3 μM	99.00%
GW768505A free base		Tie2	99.26%
CE-245677		Tie2, IC₅₀: 4.7 nM	98.00%
TIE-2/VEGFR-2 kinase-IN-1		Tie2	99.91%
RK-20448		Tie2, IC₅₀: 5.85 μM	99.38%
Regorafenib mesylate		Tie2, IC₅₀: 311 ± 46 nM
TIE-2/VEGFR-2 kinase-IN-5		Tie2, IC₅₀: 7.78 nM
Zerumin A	Tie1	Tie2
LY2457546		Tie2
TIE-2/VEGFR-2 kinase-IN-3		Tie2, IC₅₀: 6.9 nM
TIE-2/VEGFR-2 kinase-IN-4		Tie2, IC₅₀: 5.2 mM
SJ-C1044		Tie2, IC₅₀: 23 nM	98.63%
Flt-3 Inhibitor III		Tie2, IC₅₀: 8.0 μM
BSF-466895		Tie2, IC₅₀: 5 nM

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