1. GPCR/G Protein
  2. Adenosine Receptor
  3. UP202-56

UP202-56 is an adenosine analogue, which is an adenosinergic agonist.

For research use only. We do not sell to patients.

UP202-56 Chemical Structure

UP202-56 Chemical Structure

CAS No. : 163838-04-8

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Description

UP202-56 is an adenosine analogue, which is an adenosinergic agonist.

IC50 & Target

Adenosine Receptor[1][2]

In Vitro

The effects of oral administration of UP202-56, an adenosine analogue, are assessed on carrageenan-induced spinal c-Fos protein expression and peripheral oedema. Oral UP202-56 (10, 30 or 50 mg/kg) dose-dependently reduces the number of carrageenan-induced c-Fos like immunoreactivity (c-Fos-LI) neurons (r=0.931. P<0.0001), with the highest dose of UP202-56 producing 72±4% reduction of the total number of carrageenan-induced spinal c-Fos-LI neurons, and 12±3% and 33±6% of reduction of control carrageenan oedema at paw and ankle levels, respectively. UP202-56 dose-dependently reduces the spinal c-Fos protein expression in carrageenan model of inflammatory pain[1]. UP202-56 is an adenosinergic agonist[2].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

594.70

Formula

C34H38N6O4

CAS No.
SMILES

O[C@H]1[C@@H](O[C@H](C(CC2CC2)=O)[C@H]1O)N3C4=C(C(NCCC5=CN(CC6=C(C=CC(C)=C6)C)C7=C5C=C(C)C=C7)=NC=N4)N=C3

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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UP202-56 Related Classifications

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    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Product Name:
UP202-56
Cat. No.:
HY-U00226
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