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AKR1C3-IN-4 

Cat. No.: HY-138557
Handling Instructions

AKR1C3-IN-4 is a potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitor with an IC50 of 0.56 μM. AKR1C3-IN-4 has the potential for castrate resistant prostate cancer (CRPC) research.

For research use only. We do not sell to patients.

AKR1C3-IN-4 Chemical Structure

AKR1C3-IN-4 Chemical Structure

CAS No. : 1284180-11-5

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 88 In-stock
Estimated Time of Arrival: December 31
50 mg USD 80 In-stock
Estimated Time of Arrival: December 31
100 mg   Get quote  
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Based on 1 publication(s) in Google Scholar

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Description

AKR1C3-IN-4 is a potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitor with an IC50 of 0.56 μM. AKR1C3-IN-4 has the potential for castrate resistant prostate cancer (CRPC) research[1].

IC50 & Target

IC50: 0.56 μM (AKR1C3) and 15.1 μM (AKR1C2)[1]

In Vitro

AKR1C3-IN-4 has an IC50 of 15.1 μM for AKR1C2[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

281.23

Formula

C₁₄H₁₀F₃NO₂

CAS No.

1284180-11-5

SMILES

O=C(O)C1=CC=CC(NC2=CC=C(C(F)(F)F)C=C2)=C1

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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Keywords:

AKR1C3-IN-4Othersaldo-ketoreductase1C3AKR1C3castrateresistantprostatecancerCRPCAKR1C2Inhibitorinhibitorinhibit

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AKR1C3-IN-4
Cat. No.:
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