PG-911
PG-911 is a full MC5R agonist (EC50 = 0.031 nM for hMC5R). PG-911 is also a full antagonist at the hMC3R and the hMC4R (Kb: 0.38 nM and 0.17 nM, respectively). PG-911 can be used in the research of neurological disorders.
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- Formel: C53H71N13O10
- Molecular Weight:1050.21
-
Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biologische Aktivität
|
hMC5R 0.031 nM (EC50) |
hMC3R 0.38 nM (Kb) |
hMC4R 0.17 nM (Kb) |
Chemical Information
-
Molecular Weight 1050.21
-
Formel C53H71N13O10
-
Sequence
Ac-{Nle}-cyclo(Asp-{Hyp}-{d-Nal}-Arg-Trp-Lys)
-
Sequence Shortening
Ac-{Nle}-cyclo(D-{Hyp}-{d-Nal}-RWK)
-
Versand
Room temperature in continental US; may vary elsewhere.
-
Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)