BMS-948
BMS-948 is a RARβ-selective transcriptional agonist with an EC50 of 0.1 μM. BMS-948 is used in the research of tumor diseases, embryonic development and tissue remodeling.
For research use only. We do not sell to patients.
- CAS No.: 168901-49-3
- Formula: C24H17NO3
- Molecular Weight:367.40
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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RXRβ 0.1 μM (EC50) |
BMS-948 acts as a fully selective agonist of RARβ in HeLa cells, with an EC50 of 0.1 μM for RARβ-mediated transactivation, and exhibits extremely low activity against RARα and RARγ[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 168901-49-3
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Molecular Weight 367.40
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Formula C24H17NO3
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SMILES
O=C(O)C1=CC=C(C=C1)NC(=O)C2=CC=C3C=CC=C(C=4C=CC=CC4)C3=C2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)