1202916-90-2
1202916-90-2
Chemical Structure
CX-6258
- CAS No.: 1202916-90-2
- Formula:C26H24ClN3O3
- Molecular Weight:461.94
IUPAC Name: (E)-5-chloro-3-((5-(3-(4-methyl-1,4-diazepane-1-carbonyl)phenyl)furan-2-yl)methylene)indolin-2-one
InChIKey: KGBPLKOPSFDBOX-CJLVFECKSA-N
SMILES: O=C1NC2=CC=C(Cl)C=C2/C1=C\C3=CC=C(C4=CC=CC(C(N5CCCN(C)CC5)=O)=C4)O3
Biological Activity: CX-6258 is a potent and kinase selective pan-Pim kinases inhibitor, with IC50s of 5 nM, 25 nM and 16 nM for Pim-1, Pim-2 and Pim-3, respectively[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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CX-6258 | 98.06% | CX-6258 is a potent and kinase selective pan-Pim kinases inhibitor, with IC50s of 5 nM, 25 nM and 16 nM for Pim-1, Pim-2 and Pim-3, respectively. | ||||||||||||||||||||
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References
Keywords
