1265916-41-3
1265916-41-3
Chemical Structure
BIX02189
- CAS No.: 1265916-41-3
- Formula:C27H28N4O2
- Molecular Weight:440.55
IUPAC Name: (Z)-3-(((3-((dimethylamino)methyl)phenyl)amino)(phenyl)methylene)-N,N-dimethyl-2-oxoindoline-6-carboxamide
InChIKey: HOMJAAIVTDVQJA-IZHYLOQSSA-N
SMILES: O=C(N(C)C)C1=CC(NC2=O)=C(/C2=C(C3=CC=CC=C3)/NC4=CC=CC(CN(C)C)=C4)C=C1
Biological Activity: BIX02189 is a potent and selective MEK5 inhibitor with an IC50 of 1.5 nM. BIX02189 also inhibits ERK5 catalytic activity with an IC50 of 59 nM.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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BIX02189 | 99.72% | BIX02189 is a potent and selective MEK5 inhibitor with an IC50 of 1.5 nM. BIX02189 also inhibits ERK5 catalytic activity with an IC50 of 59 nM. | ||||||||||||||||||||
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Keywords
