133040-01-4
Chemical Structure
Eprosartan
Synonym(s): SKF-108566J free base
- CAS No.: 133040-01-4
- Formula:C23H24N2O4S
- Molecular Weight:424.51
IUPAC Name: (E)-4-((2-butyl-5-(2-carboxy-3-(thiophen-2-yl)prop-1-en-1-yl)-1H-imidazol-1-yl)methyl)benzoic acid
InChIKey: OROAFUQRIXKEMV-LDADJPATSA-N
SMILES: O=C(C1=CC=C(C=C1)CN2C(/C=C(CC3=CC=CS3)/C(O)=O)=CN=C2CCCC)O
Biological Activity: Eprosartan (SKF-108566J free base) is a selective, competitive, nonpeptid and orally active angiotensin II receptor antagonist, used as an antihypertensive. Eprosartan binds angiotensin II receptor with IC50s of 9.2 nM and 3.9 nM in rat and human adrenal cortical membranes, respectively [1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Eprosartan | 99.87% | Eprosartan (SKF-108566J free base) is a selective, competitive, nonpeptid and orally active angiotensin II receptor antagonist, used as an antihypertensive. Eprosartan binds angiotensin II receptor with IC50s of 9.2 nM and 3.9 nM in rat and human adrenal cortical membranes, respectively . | ||||||||||||||||||||
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Eprosartan (Standard) | ≥98% | Eprosartan (Standard) is the analytical standard of Eprosartan. This product is intended for research and analytical applications. Eprosartan (SKF-108566J free base) is a selective, competitive, nonpeptid and orally active angiotensin II receptor antagonist, used as an antihypertensive. Eprosartan binds angiotensin II receptor with IC50s of 9.2 nM and 3.9 nM in rat and human adrenal cortical membranes, respectively . | ||||||||||||||||||||
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Eprosartan-d3 | Eprosartan-d3 is the deuterium labeled Eprosartan. Eprosartan (SKF-108566J free base) is a selective, competitive, nonpeptid and orally active angiotensin II receptor antagonist, used as an antihypertensive. Eprosartan binds angiotensin II receptor with IC50s of 9.2 nM and 3.9 nM in rat and human adrenal cortical membranes, respectively . | |||||||||||||||||||||
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Eprosartan-d6 | Eprosartan-d6 is deuterated labeled Eprosartan (HY-117743). Eprosartan (SKF-108566J free base) is a selective, competitive, nonpeptid and orally active angiotensin II receptor antagonist, used as an antihypertensive. Eprosartan binds angiotensin II receptor with IC50s of 9.2 nM and 3.9 nM in rat and human adrenal cortical membranes, respectively . | |||||||||||||||||||||
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Eprosartan-d6 hydrochloride | Eprosartan-d6 hydrochloride is deuterated labeled Eprosartan. | |||||||||||||||||||||
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-
Similarity Score 0.92
HY-15834AREprosartan mesylate (Standard) -
Similarity Score 0.53
HY-105506EXP-7711 -
Similarity Score 0.50
HY-10382EXP-6803 -
Similarity Score 0.49
HY-400849Losartan impurity 14 -
Similarity Score 0.48
HY-168157TLR7 agonist 26 -
Similarity Score 0.48
HY-12765Losartan Carboxylic Acid -
Similarity Score 0.47
HY-W099762Telmisartan impurity 9 -
Similarity Score 0.47
HY-17512Losartan -
Similarity Score 0.46
HY-145885TLR7/8 agonist 6 -
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