1380672-07-0
Chemical Structure
G007-LK
- No. CAS: 1380672-07-0
- Formula:C25H16ClN7O3S
- Molecular Weight:529.96
IUPAC Name: (E)-4-(5-(2-(4-(2-chlorophenyl)-5-(5-(methylsulfonyl)pyridin-2-yl)-4H-1,2,4-triazol-3-yl)vinyl)-1,3,4-oxadiazol-2-yl)benzonitrile
InChIKey: HIWVLHPKZNBSBE-OUKQBFOZSA-N
SMILES: ClC1=C(C=CC=C1)N2C(/C=C/C3=NN=C(C4=CC=C(C#N)C=C4)O3)=NN=C2C5=CC=C(S(C)(=O)=O)C=N5
Biological Activity: G007-LK is a potent and selective inhibitor of TNKS1 and TNKS2, with IC50s of 46 nM and 25 nM, respectively.
| Referencia número | Nombre del producto | Pureza | Descripciòn | Pricing | |||||||||||||||||||
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G007-LK | 98.52% | G007-LK is a potent and selective inhibitor of TNKS1 and TNKS2, with IC50s of 46 nM and 25 nM, respectively. | ||||||||||||||||||||
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Similarity Score 0.48
HY-184437NRAS-G4-ligand-1 -
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HY-110176ASP2535 -
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HY-115952EGFR/HER2-IN-3 -
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HY-115951EGFR/HER2-IN-2 -
Similarity Score 0.44
HY-12421BET-BAY 002 -
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HY-12421BBET-BAY 002 (S enantiomer) -
Similarity Score 0.44
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