1684386-71-7
1684386-71-7
Chemical Structure
VER-246608
- CAS No.: 1684386-71-7
- Formula:C28H23ClF2N4O4
- Molecular Weight:552.96
IUPAC Name: N-(4-(2-chloro-5-methylpyrimidin-4-yl)phenyl)-N-(4-((2,2-difluoroacetamido)methyl)benzyl)-2,4-dihydroxybenzamide
InChIKey: LCGNLQSOSJFLKR-UHFFFAOYSA-N
SMILES: O=C(C1=CC=C(O)C=C1O)N(CC2=CC=C(CNC(C(F)F)=O)C=C2)C(C=C3)=CC=C3C4=NC(Cl)=NC=C4C
Biological Activity: VER-246608 is a potent and ATP-competitive inhibitor of pyruvate dehydrogenase kinase (PDK) with IC50s of 35 nM, 40 nM, 84 nM, and 91 nM for PDK-1, PDK-3, PDK-2, and PDK-4, respectively.
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VER-246608 | 99.10% | VER-246608 is a potent and ATP-competitive inhibitor of pyruvate dehydrogenase kinase (PDK) with IC50s of 35 nM, 40 nM, 84 nM, and 91 nM for PDK-1, PDK-3, PDK-2, and PDK-4, respectively. | ||||||||||||||||||||
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Keywords
