1800025-30-2
Chemical Structure
TP-020
Synonym(s): MGAT2-IN-1
- CAS No.: 1800025-30-2
- Formula:C27H21ClF5N7O3S
- Molecular Weight:654.01
IUPAC Name: N-(4-chloro-2,6-difluorophenyl)-1-(5-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl)pyrimidin-2-yl)-7-(2-oxopyrrolidin-1-yl)indoline-5-sulfonamide
InChIKey: VSZRYLHBOKTNBO-UHFFFAOYSA-N
SMILES: O=S(C1=CC2=C(N(C3=NC=C(C4=CC(C(F)(F)F)=NN4C)C=N3)CC2)C(N5C(CCC5)=O)=C1)(NC6=C(F)C=C(Cl)C=C6F)=O
Biological Activity: TP-020 (MGAT2-IN-1), a chemical probe, is an orally active inhibitor of monoacylglycerol acyltransferase (MGAT2) with IC50 of 7.8 and 2.4 nM for human and mouse MGAT2, respectively.
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TP-020 | 99.94% | TP-020 (MGAT2-IN-1), a chemical probe, is an orally active inhibitor of monoacylglycerol acyltransferase (MGAT2) with IC50 of 7.8 and 2.4 nM for human and mouse MGAT2, respectively. | ||||||||||||||||||||
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TP-020 (Standard) | ≥98% | TP-020 (Standard) (MGAT2-IN-1 (Standard)) is the analytical standard of TP-020 (HY-101857). This product is intended for research and analytical applications. TP-020 (MGAT2-IN-1), a chemical probe, is an orally active inhibitor of monoacylglycerol acyltransferase (MGAT2) with IC50 of 7.8 and 2.4 nM for human and mouse MGAT2, respectively. | ||||||||||||||||||||
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Keywords
