209481-20-9
209481-20-9
Chemical Structure
SB 271046
- CAS No.: 209481-20-9
- Formula:C20H22ClN3O3S2
- Molecular Weight:451.99
IUPAC Name: 5-chloro-N-(4-methoxy-3-(piperazin-1-yl)phenyl)-3-methylbenzo[b]thiophene-2-sulfonamide
InChIKey: LOCQRDBFWSXQQI-UHFFFAOYSA-N
SMILES: O=S(NC1=CC=C(C(N2CCNCC2)=C1)OC)(C3=C(C)C4=C(C=CC(Cl)=C4)S3)=O
Biological Activity: SB 271046 is a potent, selective, orally active and BBB-permeable 5-HT6 receptor antagonist with a pKi of 8.92-9.09. SB 271046 show >200-fold selective for the 5-HT6 receptor over other receptors, binding sites and ion channels. SB 271046 has anticonvulsant activity[1].
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SB 271046 | SB 271046 is a potent, selective, orally active and BBB-permeable 5-HT6 receptor antagonist with a pKi of 8.92-9.09. SB 271046 show >200-fold selective for the 5-HT6 receptor over other receptors, binding sites and ion channels. SB 271046 has anticonvulsant activity. | |||||||||||||||||||||
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References
Keywords
