2196245-16-4
2196245-16-4
Chemical Structure
Lp-PLA2-IN-3
- CAS No.: 2196245-16-4
- Formula:C20H13ClF3N3O3S
- Molecular Weight:467.85
IUPAC Name: 4-amino-N-(4-(4-chloro-3-(trifluoromethyl)phenoxy)-3-cyanophenyl)benzenesulfonamide
InChIKey: GADGQEKPNKSGMT-UHFFFAOYSA-N
SMILES: O=S(C1=CC=C(N)C=C1)(NC2=CC=C(OC3=CC=C(Cl)C(C(F)(F)F)=C3)C(C#N)=C2)=O
Biological Activity: Lp-PLA2-IN-3 is a potent and orally bioavailable lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor, with an IC50 of 14 nM for recombinant human Lp-PLA2 (rhLpPLA2)[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Lp-PLA2-IN-3 | 99.94% | Lp-PLA2-IN-3 is a potent and orally bioavailable lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor, with an IC50 of 14 nM for recombinant human Lp-PLA2 (rhLpPLA2). | ||||||||||||||||||||
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Structural Analogs
-
Similarity Score 0.62
HY-180572CCR2 ligand-1 -
Similarity Score 0.59
HY-153970URAT1 inhibitor 7 -
Similarity Score 0.59
HY-153971URAT1 inhibitor 8 -
Similarity Score 0.57
HY-136657SC-43 -
Similarity Score 0.57
HY-136658STAT3-IN-48 -
Similarity Score 0.55
HY-163087PT-91 -
Similarity Score 0.54
HY-179607LUF8100 -
Similarity Score 0.54
HY-147823α-Glucosidase-IN-6 -
Similarity Score 0.54
HY-W075522N,N'-(4,5-Dicyano-1,2-phenylene)bis(4-methylbenzenesulfonamide) -
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