2230475-63-3
2230475-63-3
Chemical Structure
KDM4-IN-4
- CAS No.: 2230475-63-3
- Formula:C16H23NO
- Molecular Weight:245.36
IUPAC Name: (1R,2S,3R,4S)-3-((dimethylamino)methyl)-1-phenylbicyclo[2.2.1]heptan-2-ol
InChIKey: HGNFUCJMHJYHIN-QCEMKRCNSA-N
SMILES: O[C@@H]1[C@@]2(C3=CC=CC=C3)C[C@H](CC2)[C@@H]1CN(C)C
Biological Activity: KDM4-IN-4 (compound 47) is a potent histone lysine demethylase 4 (KDM4) inhibitor with a modest affinity binding to ~80 μM for KDM4A-Tudor domain. KDM4-IN-4 can inhibit H3K4Me3 binding to the Tudor domain in cells with an EC50 value of 105 μM. KDM4-IN-4 can be used for researching anticancer[1].
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KDM4-IN-4 | KDM4-IN-4 (compound 47) is a potent histone lysine demethylase 4 (KDM4) inhibitor with a modest affinity binding to ~80 μM for KDM4A-Tudor domain. KDM4-IN-4 can inhibit H3K4Me3 binding to the Tudor domain in cells with an EC50 value of 105 μM. KDM4-IN-4 can be used for researching anticancer. | |||||||||||||||||||||
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References
Keywords
