KDM4-IN-4
KDM4-IN-4 (compound 47) is a potent histone lysine demethylase 4 (KDM4) inhibitor with a modest affinity binding to ~80 μM for KDM4A-Tudor domain. KDM4-IN-4 can inhibit H3K4Me3 binding to the Tudor domain in cells with an EC50 value of 105 μM. KDM4-IN-4 can be used for researching anticancer.
For research use only. We do not sell to patients.
- CAS No.: 2230475-63-3
- Formula: C16H23NO
- Molecular Weight:245.36
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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KDM4A-Tudor domain 80 μM (Ki) |
Chemical Information
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CAS No. 2230475-63-3
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Molecular Weight 245.36
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Formula C16H23NO
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SMILES
O[C@@H]1[C@@]2(C3=CC=CC=C3)C[C@H](CC2)[C@@H]1CN(C)C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)