2378159-28-3

PAR2 modulator-1 Chemical Structure
2378159-28-3

Chemical Structure

PAR2 modulator-1

  • CAS No.: 2378159-28-3
  • Formula:C27H41N5O5
  • Molecular Weight:515.64

InChIKey: PMKXCZFRNZTXJG-GAIPOIILSA-N

SMILES: O=C(C1=CC=CO1)N2C3N(C([C@H](C2)NC(CC(C)C)=O)=O)[C@H](C(N(C3)CC4CCNCC4)=O)CC(C)C

Biological Activity: PAR2 modulator-1 is a biased protease-activated receptor 2 (PAR2) inhibitor. PAR2 modulator-1 blocks the PAR2-dependent MAPK signaling pathway with an IC50 value of 8.5 μM, without altering the PAR2-dependent Ca2+ signaling pathway. PAR2 modulator-1 blocks pain responses induced by PAR2 agonists. PAR2 modulator-1 can be used in the research of chronic pain[1].

Cat. No. Product Name Purity Description Pricing
HY-171096 		PAR2 modulator-1 PAR2 modulator-1 is a biased protease-activated receptor 2 (PAR2) inhibitor. PAR2 modulator-1 blocks the PAR2-dependent MAPK signaling pathway with an IC50 value of 8.5 μM, without altering the PAR2-dependent Ca2+ signaling pathway. PAR2 modulator-1 blocks pain responses induced by PAR2 agonists. PAR2 modulator-1 can be used in the research of chronic pain.
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