2719793-90-3
2719793-90-3
Chemical Structure
lunresertib
Synonym(s): RP-6306
- CAS No.: 2719793-90-3
- Formula:C18H20N4O2
- Molecular Weight:324.38
IUPAC Name: 2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethyl-1H-pyrrolo[2,3-b]pyridine-3-carboxamide
InChIKey: ARBRHWRTXPWZGN-UHFFFAOYSA-N
SMILES: O=C(C1=C(N)[N@]([C@]2=C(C)C(O)=CC=C2C)C3=NC(C)=C(C)C=C31)N
Biological Activity: lunresertib (RP-6306) is a potent, selective and orally active PKMYT1 inhibitor with an IC50 of 14 nM. lunresertib shows a high degree of selectivity over other kinases in cellular binding assays. lunresertib shows anticancer effects[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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lunresertib | 99.97% | lunresertib (RP-6306) is a potent, selective and orally active PKMYT1 inhibitor with an IC50 of 14 nM. lunresertib shows a high degree of selectivity over other kinases in cellular binding assays. lunresertib shows anticancer effects. | ||||||||||||||||||||
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lunresertib (Standard) | ≥98% | lunresertib (Standard) is the analytical standard of lunresertib (HY-145817A). This product is intended for research and analytical applications. lunresertib (RP-6306) is a potent, selective and orally active PKMYT1 inhibitor with an IC50 of 14 nM. lunresertib shows a high degree of selectivity over other Kinases in cellular binding assays. lunresertib shows anticancer effects. | ||||||||||||||||||||
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Structural Analogs
-
Similarity Score 1.00
HY-145817(Rac)-lunresertib -
Similarity Score 1.00
HY-145817B(R)-lunresertib -
Similarity Score 0.81
HY-145664Myt1-IN-1 -
Similarity Score 0.70
HY-176957PKMYT1-IN-11 -
Similarity Score 0.66
HY-170517PKMYT1-IN-8 -
Similarity Score 0.65
HY-159937PKMYT1-IN-7 -
Similarity Score 0.63
HY-145666Myt1-IN-3 -
Similarity Score 0.59
HY-145665Myt1-IN-2 -
Similarity Score 0.55
HY-182906XL495 -
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