62001-32-5
62001-32-5
Chemical Structure
RSK2-IN-4
- CAS No.: 62001-32-5
- Formula:C13H11ClN4
- Molecular Weight:258.71
IUPAC Name: N-((1H-benzo[d][1,2,3]triazol-1-yl)methyl)-4-chloroaniline
InChIKey: PHAXIVPIOCGFIQ-UHFFFAOYSA-N
SMILES: ClC1=CC=C(NCN2N=NC3=C2C=CC=C3)C=C1
Biological Activity: RSK2-IN-4 (Compound 10) is a RSK2 inhibitor, with an inhibition rate of 13.73% on RSK2 activity at 10 μM. RSK2-IN-4 binds to the ATP-binding site of RSK2 in the NTKD (N-terminal kinase domain), with the electron-donating group at the 4-position of the phenyl ring being the key determinant for its inhibitory activity [1].
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RSK2-IN-4 | RSK2-IN-4 (Compound 10) is a RSK2 inhibitor, with an inhibition rate of 13.73% on RSK2 activity at 10 μM. RSK2-IN-4 binds to the ATP-binding site of RSK2 in the NTKD (N-terminal kinase domain), with the electron-donating group at the 4-position of the phenyl ring being the key determinant for its inhibitory activity . | |||||||||||||||||||||
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References
Keywords
