77779-60-3
77779-60-3
Chemical Structure
CGS 8216
- CAS No.: 77779-60-3
- Formula:C16H11N3O
- Molecular Weight:261.28
IUPAC Name: 2-phenyl-2,5-dihydro-3H-pyrazolo[4,3-c]quinolin-3-one
InChIKey: WRHJCJHWJSQAHY-UHFFFAOYSA-N
SMILES: O=C1N(C2=CC=CC=C2)N=C3C1=CNC4=C3C=CC=C4
Biological Activity: CGS 8216 is a non-benzodiazepine brain benzodiazepine receptor ligand that binds to rat forebrain membranes with high affinity and specificity. CGS 8216 also inhibits 3H-flunitrazepam (3H-FLU) binding to rat synaptosomal membranes and blocks 3H-FLU labeling of brain benzodiazepine receptors in vivo with potency equivalent to Diazepam[1].
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CGS 8216 | 99.85% | CGS 8216 is a non-benzodiazepine brain benzodiazepine receptor ligand that binds to rat forebrain membranes with high affinity and specificity. CGS 8216 also inhibits 3H-flunitrazepam (3H-FLU) binding to rat synaptosomal membranes and blocks 3H-FLU labeling of brain benzodiazepine receptors in vivo with potency equivalent to Diazepam. | ||||||||||||||||||||
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References
Keywords
