LSD1-IN-17
LSD1-IN-17 (compound 5b) is a potent LSD1 inhibitor. LSD1-IN-17 can inhibit LSD1-CoREST, MAO-A and MAO-B, with IC50 values of 0.005, 0.028, and 0.820 μM, respectively. LSD1-IN-17 displays cell growth arrest in prostate cancer LNCaP cells, with an IC50 of 17.2 μM.
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- CAS. Nr.: 3033060-70-4
- Formel: C20H18N2OS
- Molecular Weight:334.43
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biologische Aktivität
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KDM1/LSD1 |
MAO-A 0.028 ± 0. μM (IC50) |
MAO-B 0.820 ± 0. μM (IC50) |
Chemical Information
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CAS. Nr. 3033060-70-4
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Molecular Weight 334.43
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Formel C20H18N2OS
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SMILES
NC1CC1C2=CC=C(C=C2)NC(C3=CC=CC(C4=CSC=C4)=C3)=O
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)