MDA7
MDA7 is the selective agonist for cannabinoid receptor 2 with EC50 of 128 nM and 67.4 nM in human CB2 receptor and rat CB2 receptor. MDA7 exhibits good affinity to human CB2 receptor and rat CB2 receptor with Ki of 422 nM and 238 nM. MDA7 exhibits analgesic activity in rats models.
Nos produits utilisent uniquement pour la recherche. Nous ne vendons pas aux patients.
- CAS No.: 1103840-28-3
- Formule: C22H25NO2
- Masse moléculaire:335.44
-
Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
|
rat CB2-R 67.4 nM (IC50) |
hCB2-R 128 nM (IC50) |
rat CB2-R 238 nM (Ki) |
hCB2-R 422 nM (Ki) |
rCB1-R 2565 nM (Ki) |
Chemical Information
-
CAS No. 1103840-28-3
-
Masse moléculaire 335.44
-
Formule C22H25NO2
-
SMILES
O=C(N1CCCCC1)C2=CC=C3C(OCC3(CC4=CC=CC=C4)C)=C2
-
Livraison
Room temperature in continental US; may vary elsewhere.
-
Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)