1. Cell Cycle/DNA Damage
    Stem Cell/Wnt
    JAK/STAT Signaling
  2. Casein Kinase
    Pim
  3. CK2/PIM1-IN-1

CK2/PIM1-IN-1 

Cat. No.: HY-135816
Handling Instructions

CK2/PIM1-IN-1 is an inhibitor of CK2 and PIM1, with IC50s of 3.787 μM and 4.327 μM for CK2 and PIM1, respectively. CK2/PIM1-IN-1 is developed for the research of proliferative disorders such as cancer, as well as other kinase-associated conditions including inflammation, pain, vascular disorders, pathogenic infections and certain immunological disorders.

For research use only. We do not sell to patients.

CK2/PIM1-IN-1 Chemical Structure

CK2/PIM1-IN-1 Chemical Structure

CAS No. : 292640-28-9

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Description

CK2/PIM1-IN-1 is an inhibitor of CK2 and PIM1, with IC50s of 3.787 μM and 4.327 μM for CK2 and PIM1, respectively. CK2/PIM1-IN-1 is developed for the research of proliferative disorders such as cancer, as well as other kinase-associated conditions including inflammation, pain, vascular disorders, pathogenic infections and certain immunological disorders[1].

IC50 & Target

CK2

3.787 μM (IC50)

PIM1

4.327 μM (IC50)

In Vitro

CK2/PIM1-IN-1 a PIM kinases and CK2 inhibitor extracted from patent WO2010148351A1, Compound Example 64[1].

Molecular Weight

331.37

Formula

C₁₅H₉NO₄S₂

CAS No.

292640-28-9

SMILES

O=C(O)C1=CC=CC=C1C2=CC=C(/C=C(SC(N3)=S)\C3=O)O2

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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Keywords:

CK2/PIM1-IN-1Casein KinasePimPim kinasescaseinkinaseCK2PIM1kinase-associatedInhibitorinhibitorinhibit

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