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Cat. No.: HY-P3547

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(D-Met2,Pro5)-Enkephalinamide

(D-Met2,Pro5)-Enkephalinamide is a highly potent opiate agonist, and shows antinociceptive activity.

For research use only. We do not sell to patients.

CAS No.: 63307-63-1
Formula: C₃₀H₄₀N₆O₆S
Molecular Weight:612.74

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

(D-Met2,Pro5)-Enkephalinamide Chemical Structure

CAS No.: 63307-63-1

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- In Vivo
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
Classifications
Bioz

Biological Activity

Description

(D-Met2,Pro5)-Enkephalinamide is a highly potent opiate agonist, and shows antinociceptive activity^[1]^[2]^[3].

All Opioid Receptor Isoforms :

In Vivo

(D-Met2,Pro5)-Enkephalinamide (intravenous injection; 0.25 and 0.5 mg/kg; once) leads to the decreasement of prolactin (PRL) secretion in lactating rats^[2].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model:

Wistar lactating rats^[2]
Dosage:

0.25 and 0.5 mg/kg
Administration:

Intravenous injection; 0.25 and 0.5 mg/kg; once
Result:

Decreased plasma PRL levels 15 min after the administration in continuously lactating rats.
Produced a marked depression in plasma PRL concentration in non-deprived lactating mothers.

Chemical Information

CAS No. 63307-63-1
Molecular Weight 612.74
Formula C₃₀H₄₀N₆O₆S
Sequence Shortening

Y-{d-Met}-GFP-NH2
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (271 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Decsi L, et al. Effect of (D-Met2, Pro5)enkephalinamide, a highly potent opiate agonist, on the drinking behaviour of rats. Neuropharmacology. 1985 Jan;24(1):5-8. [Content Brief]

[2]. Nagy G, et al. (D-Met2,Pro5) enkephalinamide causes a decrease in plasma prolactin levels of lactating rats continuously suckled and an increase in those deprived of their litter. Regul Pept. 1984 Jul;8(4):321-6. [Content Brief]

[3]. Wollemann M, et al. Effect of Met-enkephalin and (D-Met2,Pro5)-enkephalinamide on the adenylate cyclase activity of rat brain. Neurochem Res. 1979 Oct;4(5):627-31. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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Biological Activity
- Description
- In Vivo
Chemical Information
Purity & Documentation
References

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(D-Met2,Pro5)-Enkephalinamide

All Opioid Receptor Isoforms

Biological Activity

Chemical Information

Purity & Documentation

References

Calculators

Help & FAQs

(D-Met2,Pro5)-Enkephalinamide Related Classifications

HY-P3547 Related Classifications