Dopamine D2 receptor antagonist-3
Dopamine D2 receptor antagonist-3 (Example 17) is an orally active and selective dopamine D2 receptor antagonist with a pIC50 of 5.52. Dopamine D2 receptor antagonist-3 exhibits antipsychotic activity in the Apomorphine (HY-12723) induced agitation in rats. Dopamine D2 receptor antagonist-3 can be used for psychiatric and neurological disorders research.
For research use only. We do not sell to patients.
- CAS No.: 1032714-06-9
- Formula: C18H17F4N5
- Molecular Weight:379.35
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Dopamine Receptor Isoforms
More
Biological Activity
|
D2 Receptor 5.52 (pIC50) |
Chemical Information
-
CAS No. 1032714-06-9
-
Molecular Weight 379.35
-
Formula C18H17F4N5
-
SMILES
FC1=CC(CN2CCC(NC3=NN=C(C#N)C=C3)CC2)=CC(C(F)(F)F)=C1
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)