Picenadol
Picenadol (LY-150720) is an opioid mixed agonist-antagonist analgesic. Picenadol is an external racemic mixture, where its d-isomer (LY136596) is a potent μ-opioid receptor agonist, and the l-isomer (LY136595) is a weak μ-receptor competitive antagonist, which can inhibit the agonist effect and reduce the risk of dependence. Picenadol has anticholinergic activity.
For research use only. We do not sell to patients.
- CAS No.: 79201-85-7
- Formula: C16H25NO
- Molecular Weight:247.38
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Biological Activity
-
Chemical Information
- Purity & Documentation
- References
-
Help & FAQs
All Opioid Receptor Isoforms
More
Biological Activity
|
μ Opioid Receptor/MOR |
Chemical Information
-
CAS No. 79201-85-7
-
Molecular Weight 247.38
-
Formula C16H25NO
-
SMILES
CCC[C@]1([C@@H](C)CN(CC1)C)C2=CC(O)=CC=C2
-
Synonyms
LY-150720
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
[1]. Carter RB, et al. Effects of LY150720 (picenadol), a novel mixed-action opioid, on schedule-controlled responding in the squirrel monkey. Pharmacol Biochem Behav. 1984 Nov;21(5):779-86. [Content Brief]
[2]. Zimmerman DM, et al. Picenadol. Drug Alcohol Depend. 1985 Feb;14(3-4):381-401. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Picenadol Related Classifications
HY-106601 Related Classifications
Powered by Bioz